IADR Abstract Archives

Development  of Drugs for Local Treatment of Common Oral Conditions

Objective: There is a recognised need to develop topical preparations for treating common oral mucosal diseases.  Objectives: These studies aimed to develop pharmaceutical preparations that could  help treat  some oral  mucosal conditions  including  aphthous ulceration, denture stomatitis and  herpes  labialis.  Two main active ingredients were evaluated: i) low-dose doxycycline, as an active inhibitor of matrix metalloproteinases,   and ii) monocaprin,  a  1-monoglyceride of capric acid, that is virucidal against Herpes simplex and has good anti-Candidal activity.

Method: Methods: Laboratory studies tested  hydrogels  and  denture  adhesives to  deliver the active  ingredients  to  the  oral  mucosa. Clinical  trials were then  carried  out.   Recurrent oral ulcers were treated with a low dose-doxycycline (1.5 mg/g) hydrogel applied to the aphthous ulcer 4 times per day for 3 days.  A denture adhesive containing 3% monocaprin was tested in  elderly subjects to  determine its inhibition of Candida growth on the oral  mucosa and its potential use as a denture disinfectant. The anti-viral activity of monocaprin combined  with the matrix metalloproteinase inhibiting  activity of doxycycline in a muco-adhesive gel was tested in a double-blind placebo-controlled clinical trial for treating herpes labialis

Result: Results:  The results of clinical trials showed that 70% of topically treated aphthous ulcers healed by the third day compared with 25% of placebo controls (p<0.005).  The combination of monocaprin and doxycycline reduced  the healing time of herpes  labialis lesions, both at prodromal and vesicle stages, by about 2 days (p<0.05). Pain scores were also reduced. Monocaprin in a denture adhesive reduced  counts of Candida on the  oral  mucosa  but especially  on the  denture fitting  surface and had a potential for preventing oral candidosis over a longer period. 

Conclusion: Conclusion: The results indicated that the treatments of these common conditions in the oral cavity can  be  improved using topical delivery systems containing monocaprin and low-dose doxycycline.

Division: Pan European Region Meeting
Meeting: 2014 Pan European Region Meeting (Dubrovnik, Croatia)
Location: Dubrovnik, Croatia
Year: 2014
Final Presentation ID: 452
Abstract Category|Abstract Category(s): Scientific Groups
Authors
  • Holbrook, W. Peter  ( University of Iceland, Reykjavik, N/A, Iceland )
  • Kristmundsdóttir, Thordis  ( University of Iceland, Reykjavik, N/A, Iceland )
  • Thormar, Halldor  ( University of Iceland, Reykjavík, N/A, Iceland )
  • Skúlason, Skúli  ( Medis ehf., Hafnarfjordur, , Iceland )
  • SESSION INFORMATION
    Poster Session
    Pharmacology/Therapeutics/Toxicology
    09/12/2014