IADR Abstract Archives

Sequential Menaquinone And Risedronate rescue cottical bone in inactive rat

Objectives: Risedronate, an amino bisphosphonate, is a potent first-choice drug for osteoporosis. We have reported that Vitamin K2 (MK-4) administration followed by risedronate is a most effective combinatory method much superior to the administration of the two drugs together1). It was also reported that it exhibits much better effect with exercise. To prevent unnecessary side effects such as osteonecrosis of the jaw or atypical fractures of femur, we hypothesized that prior treatment with MK-4 during disuse followed by risedronate administration is an effective method to make bisphosphonate less hazardous.

Methods: Retired breeder female Wistar rats were ovariectomyzed and fed either with or without 100μg/kg/day MK-4. Half of the rats (inactive groups) were kept in small cages, which prevent rats from walking2). After 21 weeks, all the rats were returned to regular cages and treated with 1.76 mg/Kg risedronate orally once a week for 18weeks.

Results: Compared to those of femoral cortical bone of the sham-operated rats, values by nano-indentation and confocal laser Raman microspectroscopy parameters such as mineral/matrix showed significant improvement from that of inactive group by the prior MK-4 treatment.

Conclusions: Bed rest patients, if treated with MK-4 during hospitalization, may react better to later risedronate administration, which results in more resilient bone of better quality.

1)Y Matsumoto, Y Mikuni-Takagaki, Y Kozai, K Miyagawa, K Naruse, H Wakao, R Kawamata, I Kashima, T Sakurai Prior treatment with vitamin K2significantly improves the efficacy of risedronate. Osteoporos Int. 20:1863, 2009

2) K Miyagawa,Y Kozai, Y Ito, T Furuhama,K Naruse,K Nonaka, Y Nagai, H Yamato, IKashima, K Ohya,K Aoki, and Y Mikuni-TakagakiA novel underuse model shows that inactivity but not ovariectomy determines the deteriorated material properties and geometry of cortical bone in the tibia of adult rats. J.Bone  Miner. Metab. 29:422, 2011

Division: Japanese Division Meeting
Meeting: 2012 Japanese Division Meeting (Niigata, Japan)
Location: Niigata, Japan
Year: 2012
Final Presentation ID:
Abstract Category|Abstract Category(s): Scientific Program
Authors
  • Funayama, Yuta  ( Kanagawa Dental College, Yokosuka, N/A, Japan )
  • Tanaka, Takahiro  ( Kanagawa Dental College, Yokosuka, N/A, Japan )
  • Teranaka, Toshio  ( Kanagawa Dental College, Kanagawa, N/A, Japan )
  • Mikuni-takagaki, Yuko  ( Kanagawa Dental College, Yokosuka, N/A, Japan )
  • SESSION INFORMATION
    Mineralized Tissue